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Target
Sphingosine 1-phosphate receptor 2
Ligand
BDBM41655
Substrate
n/a
Meas. Tech.
Counter screen for S1P2 Agonists: Dose Response High Throughput Cell-Based Screen to Identify Activators of CRE-BLA
EC50
>50000±n/a nM
Citation
 PubChem, PC Counter screen for S1P2 Agonists: Dose Response High Throughput Cell-Based Screen to Identify Activators of CRE-BLA PubChem Bioassay (2007)[AID] 
Target
Name:
Sphingosine 1-phosphate receptor 2
Synonyms:
EDG5 | S1P2 | S1PR2 | S1PR2_HUMAN | Sphingosine 1-phosphate receptor | Sphingosine 1-phosphate receptor Edg-5 | Sphingosine-1-phosphate receptor 2 | ndothelial differentiation G-protein coupled receptor 5
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
38883.16
Organism:
Homo sapiens (Human)
Description:
Membranes isolated from S1P2-transfected CHO cells were used in ligand binding assay.
Residue:
353
Sequence:
MGSLYSEYLNPNKVQEHYNYTKETLETQETTSRQVASAFIVILCCAIVVENLLVLIAVARNSKFHSAMYLFLGNLAASDLLAGVAFVANTLLSGSVTLRLTPVQWFAREGSAFITLSASVFSLLAIAIERHVAIAKVKLYGSDKSCRMLLLIGASWLISLVLGGLPILGWNCLGHLEACSTVLPLYAKHYVLCVVTIFSIILLAIVALYVRIYCVVRSSHADMAAPQTLALLKTVTIVLGVFIVCWLPAFSILLLDYACPVHSCPILYKAHYFFAVSTLNSLLNPVIYTWRSRDLRREVLRPLQCWRPGVGVQGRRRGGTPGHHLLPLRSSSSLERGMHMPTSPTFLEGNTVV
  
Inhibitor
Name:
BDBM41655
Synonyms:
(4E)-4-(2-furanylmethylidene)-2-phenyl-5-thiazolone | (4E)-4-(2-furfurylidene)-2-phenyl-2-thiazolin-5-one | (4E)-4-(2-furylmethylene)-2-phenyl-1,3-thiazol-5(4H)-one | (4E)-4-(furan-2-ylmethylidene)-2-phenyl-1,3-thiazol-5-one | MLS000088479 | SMR000024099 | cid_5771471
Type:
Small organic molecule
Emp. Form.:
C14H9NO2S
Mol. Mass.:
255.292
SMILES:
O=C1SC(=N\C1=C\c1ccco1)c1ccccc1 |c:3|
Structure:
Search PDB for entries with ligand similarity: