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Target
Procathepsin L
Ligand
BDBM41174
Substrate
n/a
Meas. Tech.
Cathepsin L dose-response testing in the presence of cysteine
IC50
>50000±0 nM
Citation
 PubChem, PC Cathepsin L dose-response testing in the presence of cysteine PubChem Bioassay (2009)[AID] 
Target
Name:
Procathepsin L
Synonyms:
CATL1_HUMAN | CTSL | CTSL CTSL1 | CTSL1 | Cathepsin L | Cathepsin L1 | Cathepsin L1 heavy chain | Cathepsin L1 light chain | MEP | Major excreted protein | cathepsin L preproprotein
Type:
Enzyme
Mol. Mass.:
37557.19
Organism:
Homo sapiens (Human)
Description:
Purchased from Calbiochem (San Diego, CA).
Residue:
333
Sequence:
MNPTLILAAFCLGIASATLTFDHSLEAQWTKWKAMHNRLYGMNEEGWRRAVWEKNMKMIELHNQEYREGKHSFTMAMNAFGDMTSEEFRQVMNGFQNRKPRKGKVFQEPLFYEAPRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESTESDNNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV
  
Inhibitor
Name:
BDBM41174
Synonyms:
4-[[4-(morpholinomethyl)benzoyl]amino]benzoic acid methyl ester | 4-[[[4-(4-morpholinylmethyl)phenyl]-oxomethyl]amino]benzoic acid methyl ester | MLS000064549 | SMR000077137 | cid_2211303 | methyl 4-[[4-(morpholin-4-ylmethyl)benzoyl]amino]benzoate | methyl 4-[[4-(morpholin-4-ylmethyl)phenyl]carbonylamino]benzoate | methyl 4-{[4-(4-morpholinylmethyl)benzoyl]amino}benzoate
Type:
Small organic molecule
Emp. Form.:
C20H22N2O4
Mol. Mass.:
354.3997
SMILES:
COC(=O)c1ccc(NC(=O)c2ccc(CN3CCOCC3)cc2)cc1
Structure:
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