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Target
Regulator of G-protein signaling 16
Ligand
BDBM47810
Substrate
n/a
Meas. Tech.
Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao.
EC50
>30000±n/a nM
Citation
 PubChem, PC Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao. PubChem Bioassay (2009)[AID] 
Target
Name:
Regulator of G-protein signaling 16
Synonyms:
RGS16 | RGS16_HUMAN | RGSR | Regulator of G-protein signaling 16 (RGS16) | regulator of G-protein signalling 16
Type:
Enzyme Catalytic Domain
Mol. Mass.:
22748.87
Organism:
Homo sapiens (Human)
Description:
gi_156416009
Residue:
202
Sequence:
MCRTLAAFPTTCLERAKEFKTRLGIFLHKSELGCDTGSTGKFEWGSKHSKENRNFSEDVLGWRESFDLLLSSKNGVAAFHAFLKTEFSEENLEFWLACEEFKKIRSATKLASRAHQIFEEFICSEAPKEVNIDHETHELTRMNLQTATATCFDAAQGKTRTLMEKDSYPRFLKSPAYRDLAAQASAASATLSSCSLDEPSHT
  
Inhibitor
Name:
BDBM47810
Synonyms:
2-(pyridin-4-ylcarbonylamino)ethyl N-(3,4-dichlorophenyl)carbamate | 2-(pyridine-4-carbonylamino)ethyl N-(3,4-dichlorophenyl)carbamate | MLS001034017 | N-(3,4-dichlorophenyl)carbamic acid 2-[[oxo(pyridin-4-yl)methyl]amino]ethyl ester | N-(3,4-dichlorophenyl)carbamic acid 2-isonicotinamidoethyl ester | SMR000385849 | cid_2121675
Type:
Small organic molecule
Emp. Form.:
C15H13Cl2N3O3
Mol. Mass.:
354.188
SMILES:
Clc1ccc(NC(=O)OCCNC(=O)c2ccncc2)cc1Cl
Structure:
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