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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM31999
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
2020±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM31999
Synonyms:
3-[5-(4-Ethyl-phenyl)-tetrazol-2-yl]-propionic acid methyl ester | 3-[5-(4-ethylphenyl)-2-tetrazolyl]propanoic acid methyl ester | 3-[5-(4-ethylphenyl)tetrazol-2-yl]propionic acid methyl ester | MLS000029758 | SMR000002517 | cid_647427 | methyl 3-[5-(4-ethylphenyl)-1,2,3,4-tetrazol-2-yl]propanoate | methyl 3-[5-(4-ethylphenyl)tetrazol-2-yl]propanoate
Type:
Small organic molecule
Emp. Form.:
C13H16N4O2
Mol. Mass.:
260.2917
SMILES:
CCc1ccc(cc1)-c1nnn(CCC(=O)OC)n1
Structure:
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