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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48110
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
6270±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48110
Synonyms:
MLS000035103 | N-[6-(2-methylpropanoylamino)pyridin-3-yl]pyridine-2-carboxamide | N-[6-(isobutyrylamino)-3-pyridyl]picolinamide | N-[6-[(2-methyl-1-oxopropyl)amino]-3-pyridinyl]-2-pyridinecarboxamide | Pyridine-2-carboxylic acid (6-isobutyrylamino-pyridin-3-yl)-amide | SMR000005528 | cid_649501
Type:
Small organic molecule
Emp. Form.:
C15H16N4O2
Mol. Mass.:
284.3131
SMILES:
CC(C)C(=O)Nc1ccc(NC(=O)c2ccccn2)cn1
Structure:
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