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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48114
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
9010±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48114
Synonyms:
MLS000035120 | N-[6-(2-furoylamino)-3-pyridyl]picolinamide | N-[6-(furan-2-carbonylamino)pyridin-3-yl]pyridine-2-carboxamide | N-[6-(furan-2-ylcarbonylamino)pyridin-3-yl]pyridine-2-carboxamide | N-[6-[[2-furanyl(oxo)methyl]amino]-3-pyridinyl]-2-pyridinecarboxamide | Pyridine-2-carboxylic acid {6-[(furan-2-carbonyl)-amino]-pyridin-3-yl}-amide | SMR000005518 | cid_655025
Type:
Small organic molecule
Emp. Form.:
C16H12N4O3
Mol. Mass.:
308.2915
SMILES:
O=C(Nc1ccc(NC(=O)c2ccccn2)cn1)c1ccco1
Structure:
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