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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM40577
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
26500±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM40577
Synonyms:
4-(4-Pyrrolidin-1-yl-quinazolin-2-ylamino)-phenol | 4-[(4-pyrrolidin-1-ylquinazolin-2-yl)amino]phenol;hydrochloride | 4-[(4-pyrrolidinoquinazolin-2-yl)amino]phenol;hydrochloride | 4-[[4-(1-pyrrolidinyl)-2-quinazolinyl]amino]phenol;hydrochloride | MLS000026828 | SMR000013024 | cid_6602552
Type:
Small organic molecule
Emp. Form.:
C18H18N4O
Mol. Mass.:
306.3617
SMILES:
Oc1ccc(Nc2nc(N3CCCC3)c3ccccc3n2)cc1
Structure:
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