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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM34247
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
4200±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM34247
Synonyms:
3,6-bis(2-pyridinyl)pyridazine | 3,6-bis(2-pyridyl)pyridazine | 3,6-dipyridin-2-ylpyridazine | MLS000038780 | SMR000036841 | cid_659563
Type:
Small organic molecule
Emp. Form.:
C14H10N4
Mol. Mass.:
234.256
SMILES:
c1ccc(nc1)-c1ccc(nn1)-c1ccccn1
Structure:
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