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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48120
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
8500±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48120
Synonyms:
1-(4-methoxyphenyl)-N-prop-2-enyl-4-pyrazolo[3,4-d]pyrimidinamine | 1-(4-methoxyphenyl)-N-prop-2-enyl-pyrazolo[3,4-d]pyrimidin-4-amine | 1-(4-methoxyphenyl)-N-prop-2-enylpyrazolo[3,4-d]pyrimidin-4-amine | MLS000036778 | SMR000035743 | allyl-[1-(4-methoxyphenyl)pyrazolo[3,4-d]pyrimidin-4-yl]amine | cid_661248
Type:
Small organic molecule
Emp. Form.:
C15H15N5O
Mol. Mass.:
281.3125
SMILES:
COc1ccc(cc1)-n1ncc2c(NCC=C)ncnc12
Structure:
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