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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48123
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
2680±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48123
Synonyms:
2-(2,4-dimethylphenyl)-1,3-benzoxazol-5-amine | MLS000040469 | SMR000045362 | [2-(2,4-dimethylphenyl)-1,3-benzoxazol-5-yl]amine | cid_664476
Type:
Small organic molecule
Emp. Form.:
C15H14N2O
Mol. Mass.:
238.2845
SMILES:
Cc1ccc(-c2nc3cc(N)ccc3o2)c(C)c1
Structure:
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