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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48127
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
8020±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48127
Synonyms:
3-([1,2,4]triazolo[3,4-b][1,3]benzothiazol-1-ylsulfanylmethyl)-1,2,3-benzotriazin-4-one | 3-[([1,2,4]triazolo[3,4-b][1,3]benzothiazol-1-ylthio)methyl]-1,2,3-benzotriazin-4-one | MLS000056046 | SMR000067124 | cid_2128690
Type:
Small organic molecule
Emp. Form.:
C16H10N6OS2
Mol. Mass.:
366.42
SMILES:
O=c1n(CSc2nnc3sc4ccccc4n23)nnc2ccccc12
Structure:
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