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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48129
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
13200±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48129
Synonyms:
4-[2,5-dimethyl-1-(2-phenylethyl)-3-pyrrolyl]-2-thiazolamine;hydrochloride | 4-[2,5-dimethyl-1-(2-phenylethyl)pyrrol-3-yl]-1,3-thiazol-2-amine;hydrochloride | MLS000056022 | SMR000068520 | [4-(2,5-dimethyl-1-phenethyl-pyrrol-3-yl)thiazol-2-yl]amine;hydrochloride | cid_6602929
Type:
Small organic molecule
Emp. Form.:
C17H19N3S
Mol. Mass.:
297.418
SMILES:
Cc1cc(-c2csc(N)n2)c(C)n1CCc1ccccc1
Structure:
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