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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48130
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
12100±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48130
Synonyms:
2-[(3-chloranylimidazo[1,2-a]pyridin-2-yl)methylsulfanyl]-1,3-benzoxazole | 2-[(3-chloro-2-imidazo[1,2-a]pyridinyl)methylthio]-1,3-benzoxazole | 2-[(3-chloroimidazo[1,2-a]pyridin-2-yl)methylsulfanyl]-1,3-benzoxazole | 2-[(3-chloroimidazo[1,2-a]pyridin-2-yl)methylthio]-1,3-benzoxazole | MLS000097840 | SMR000059985 | cid_914513
Type:
Small organic molecule
Emp. Form.:
C15H10ClN3OS
Mol. Mass.:
315.777
SMILES:
Clc1c(CSc2nc3ccccc3o2)nc2ccccn12
Structure:
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