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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48132
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
1820±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48132
Synonyms:
MLS000055504 | N-(3-imidazol-1-ylpropyl)-2-[(2,3,5,6-tetramethylphenyl)sulfonylamino]benzamide;hydrochloride | N-[3-(1-imidazolyl)propyl]-2-[(2,3,5,6-tetramethylphenyl)sulfonylamino]benzamide;hydrochloride | SMR000066013 | cid_6602839
Type:
Small organic molecule
Emp. Form.:
C23H28N4O3S
Mol. Mass.:
440.558
SMILES:
Cc1cc(C)c(C)c(c1C)S(=O)(=O)Nc1ccccc1C(=O)NCCCn1ccnc1
Structure:
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