Reaction Details Report a problem with these data
Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48133
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
12300±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48133
Synonyms:
2-methyl-6-phenyl-imidazo[2,1-b][1,3,4]thiadiazole | 2-methyl-6-phenylimidazo[2,1-b][1,3,4]thiadiazole | MLS000097928 | SMR000060563 | cid_3000039
Type:
Small organic molecule
Emp. Form.:
C11H9N3S
Mol. Mass.:
215.274
SMILES:
Cc1nn2cc(nc2s1)-c1ccccc1
Structure:
Search PDB for entries with ligand similarity: