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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM38963
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
6940±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM38963
Synonyms:
5-(benzoxymethyl)-7-(piperidinomethyl)quinolin-8-ol | 5-(phenylmethoxymethyl)-7-(1-piperidinylmethyl)-8-quinolinol | 5-(phenylmethoxymethyl)-7-(piperidin-1-ylmethyl)quinolin-8-ol | MLS000094939 | SMR000030493 | cid_3238417
Type:
Small organic molecule
Emp. Form.:
C23H26N2O2
Mol. Mass.:
362.4647
SMILES:
Oc1c(CN2CCCCC2)cc(COCc2ccccc2)c2cccnc12
Structure:
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