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Target
D(1B) dopamine receptor
Ligand
BDBM48934
Substrate
n/a
Meas. Tech.
Allosteric Modulators of D1 Receptors: Dose-dependent Counterscreen
EC50
0.0128±n/a nM
Citation
 PubChem, PC Allosteric Modulators of D1 Receptors: Dose-dependent Counterscreen PubChem Bioassay (2007)[AID] 
Target
Name:
D(1B) dopamine receptor
Synonyms:
D(5) dopamine receptor | D1beta dopamine receptor | DOPAMINE D5 | DRD1B | DRD1L2 | DRD5 | DRD5_HUMAN | dopamine receptor D5
Type:
Protein
Mol. Mass.:
52943.41
Organism:
Homo sapiens (Human)
Description:
P21918
Residue:
477
Sequence:
MLPPGSNGTAYPGQFALYQQLAQGNAVGGSAGAPPLGPSQVVTACLLTLLIIWTLLGNVLVCAAIVRSRHLRANMTNVFIVSLAVSDLFVALLVMPWKAVAEVAGYWPFGAFCDVWVAFDIMCSTASILNLCVISVDRYWAISRPFRYKRKMTQRMALVMVGLAWTLSILISFIPVQLNWHRDQAASWGGLDLPNNLANWTPWEEDFWEPDVNAENCDSSLNRTYAISSSLISFYIPVAIMIVTYTRIYRIAQVQIRRISSLERAAEHAQSCRSSAACAPDTSLRASIKKETKVLKTLSVIMGVFVCCWLPFFILNCMVPFCSGHPEGPPAGFPCVSETTFDVFVWFGWANSSLNPVIYAFNADFQKVFAQLLGCSHFCSRTPVETVNISNELISYNQDIVFHKEIAAAYIHMMPNAVTPGNREVDNDEEEGPFDRMFQIYQTSPDGDPVAESVWELDCEGEISLDKITPFTPNGFH
  
Inhibitor
Name:
BDBM48934
Synonyms:
4-(4-bromophenyl)-4,10-dihydro-[1,3,5]triazino[1,2-a]benzimidazol-2-amine;ethanoic acid | MLS000048687 | SMR000060236 | acetic acid;4-(4-bromophenyl)-4,10-dihydro-[1,3,5]triazino[1,2-a]benzimidazol-2-amine | acetic acid;[4-(4-bromophenyl)-4,10-dihydro-[1,3,5]triazino[1,2-a]benzimidazol-2-yl]amine | cid_5742515
Type:
Small organic molecule
Emp. Form.:
C15H12BrN5
Mol. Mass.:
342.193
SMILES:
NC1=NC(c2ccc(Br)cc2)n2c(N1)nc1ccccc21 |t:1|
Structure:
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