Reaction Details Report a problem with these data
Target
POsterior Segregation
Ligand
BDBM33071
Substrate
n/a
Meas. Tech.
Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA
EC50
300000±n/a nM
Citation
 PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA PubChem Bioassay (2009)[AID] 
Target
Name:
POsterior Segregation
Synonyms:
POsterior Segregation family member (pos-1)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
29838.90
Organism:
Caenorhabditis elegans
Description:
gi_17562800
Residue:
264
Sequence:
MADNDFLSGEAIMVFKKEILDSHSDFTRSLSHQSASPEAYDQENVFSQDFQPFMKQDKETQNSASQPTSEQSLANRDPCTVPDDLREEMMRQRRKEDAFKTALCDAYKRSQACSYGDQCRFAHGVHELRLPMNPRGRNHPKYKTVLCDKFSMTGNCKYGTRCQFIHKIVDGNAAKLASGAHANTSSKSPARNAAAHNHSLFVPQGSTDRSMDLNQSLPIRQSDLVRAFARATRLDVSGYNSTAQLAQYFESQFQRIQQLSSHHH
  
Inhibitor
Name:
BDBM33071
Synonyms:
2,3-Di-furan-2-yl-quinoxaline-6-carboxylic acid (2-hydroxy-ethyl)-amide | 2,3-bis(2-furanyl)-N-(2-hydroxyethyl)-6-quinoxalinecarboxamide | 2,3-bis(2-furyl)-N-(2-hydroxyethyl)quinoxaline-6-carboxamide | 2,3-bis(furan-2-yl)-N-(2-hydroxyethyl)quinoxaline-6-carboxamide | MLS000529296 | SMR000121771 | cid_3157644
Type:
Small organic molecule
Emp. Form.:
C19H15N3O4
Mol. Mass.:
349.3401
SMILES:
OCCNC(=O)c1ccc2nc(-c3ccco3)c(nc2c1)-c1ccco1
Structure:
Search PDB for entries with ligand similarity: