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Target
Kallikrein-5
Ligand
BDBM49570
Substrate
n/a
Meas. Tech.
Kallikrein 5 1536 HTS Dose Response Confirmation
IC50
50000±n/a nM
Citation
 PubChem, PC Kallikrein 5 1536 HTS Dose Response Confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Kallikrein-5
Synonyms:
KLK5 | KLK5_HUMAN | Kallikrein 5 | SCTE | kallikrein-related peptidase 5 preproprotein
Type:
PROTEIN
Mol. Mass.:
32031.72
Organism:
Homo sapiens (Human)
Description:
EBI_12584
Residue:
293
Sequence:
MATARPPWMWVLCALITALLLGVTEHVLANNDVSCDHPSNTVPSGSNQDLGAGAGEDARSDDSSSRIINGSDCDMHTQPWQAALLLRPNQLYCGAVLVHPQWLLTAAHCRKKVFRVRLGHYSLSPVYESGQQMFQGVKSIPHPGYSHPGHSNDLMLIKLNRRIRPTKDVRPINVSSHCPSAGTKCLVSGWGTTKSPQVHFPKVLQCLNISVLSQKRCEDAYPRQIDDTMFCAGDKAGRDSCQGDSGGPVVCNGSLQGLVSWGDYPCARPNRPGVYTNLCKFTKWIQETIQANS
  
Inhibitor
Name:
BDBM49570
Synonyms:
5-(4-chloranyl-2-nitro-phenyl)-3-phenyl-1,2,4-oxadiazole | 5-(4-chloro-2-nitro-phenyl)-3-phenyl-1,2,4-oxadiazole | 5-(4-chloro-2-nitrophenyl)-3-phenyl-1,2,4-oxadiazole | MLS000578496 | SMR000198496 | cid_891545
Type:
Small organic molecule
Emp. Form.:
C14H8ClN3O3
Mol. Mass.:
301.685
SMILES:
[O-][N+](=O)c1cc(Cl)ccc1-c1nc(no1)-c1ccccc1
Structure:
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