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Target
Kallikrein-5
Ligand
BDBM56637
Substrate
n/a
Meas. Tech.
Kallikrein 5 1536 HTS Dose Response Confirmation
IC50
50000±n/a nM
Citation
 PubChem, PC Kallikrein 5 1536 HTS Dose Response Confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Kallikrein-5
Synonyms:
KLK5 | KLK5_HUMAN | Kallikrein 5 | SCTE | kallikrein-related peptidase 5 preproprotein
Type:
PROTEIN
Mol. Mass.:
32031.72
Organism:
Homo sapiens (Human)
Description:
EBI_12584
Residue:
293
Sequence:
MATARPPWMWVLCALITALLLGVTEHVLANNDVSCDHPSNTVPSGSNQDLGAGAGEDARSDDSSSRIINGSDCDMHTQPWQAALLLRPNQLYCGAVLVHPQWLLTAAHCRKKVFRVRLGHYSLSPVYESGQQMFQGVKSIPHPGYSHPGHSNDLMLIKLNRRIRPTKDVRPINVSSHCPSAGTKCLVSGWGTTKSPQVHFPKVLQCLNISVLSQKRCEDAYPRQIDDTMFCAGDKAGRDSCQGDSGGPVVCNGSLQGLVSWGDYPCARPNRPGVYTNLCKFTKWIQETIQANS
  
Inhibitor
Name:
BDBM56637
Synonyms:
4-methyl-N-[methyl(propyl)--sulfanylidene]benzenesulfonamide | 4-methyl-N-[methyl(propyl)-lambda~4~-sulfanylidene]benzenesulfonamide | 4-methyl-N-[methyl(propyl)sulfuranylidene]benzenesulfonamide | MLS000704720 | SMR000231807 | cid_3041266
Type:
Small organic molecule
Emp. Form.:
C11H17NO2S2
Mol. Mass.:
259.388
SMILES:
CCC=S(C)NS(=O)(=O)c1ccc(C)cc1 |w:2.1|
Structure:
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