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Target
Kallikrein-5
Ligand
BDBM56803
Substrate
n/a
Meas. Tech.
Kallikrein 5 1536 HTS Dose Response Confirmation
IC50
50000±n/a nM
Citation
 PubChem, PC Kallikrein 5 1536 HTS Dose Response Confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Kallikrein-5
Synonyms:
KLK5 | KLK5_HUMAN | Kallikrein 5 | SCTE | kallikrein-related peptidase 5 preproprotein
Type:
PROTEIN
Mol. Mass.:
32031.72
Organism:
Homo sapiens (Human)
Description:
EBI_12584
Residue:
293
Sequence:
MATARPPWMWVLCALITALLLGVTEHVLANNDVSCDHPSNTVPSGSNQDLGAGAGEDARSDDSSSRIINGSDCDMHTQPWQAALLLRPNQLYCGAVLVHPQWLLTAAHCRKKVFRVRLGHYSLSPVYESGQQMFQGVKSIPHPGYSHPGHSNDLMLIKLNRRIRPTKDVRPINVSSHCPSAGTKCLVSGWGTTKSPQVHFPKVLQCLNISVLSQKRCEDAYPRQIDDTMFCAGDKAGRDSCQGDSGGPVVCNGSLQGLVSWGDYPCARPNRPGVYTNLCKFTKWIQETIQANS
  
Inhibitor
Name:
BDBM56803
Synonyms:
3-[(2,4-dichlorophenyl)carbamoylamino]benzoic acid methyl ester | 3-[[(2,4-dichloroanilino)-oxomethyl]amino]benzoic acid methyl ester | MLS000851404 | SMR000457847 | cid_2806337 | methyl 3-[(2,4-dichlorophenyl)carbamoylamino]benzoate | methyl 3-{[(2,4-dichloroanilino)carbonyl]amino}benzoate
Type:
Small organic molecule
Emp. Form.:
C15H12Cl2N2O3
Mol. Mass.:
339.173
SMILES:
COC(=O)c1cccc(NC(=O)Nc2ccc(Cl)cc2Cl)c1
Structure:
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