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Target
Tubulin polymerization-promoting protein
Ligand
BDBM59225
Substrate
n/a
Meas. Tech.
Tubulin Polymerization
IC50
1.5e+3± 2e+2 nM
Citation
Kong, Y; Grembecka, J; Edler, MC; Hamel, E; Mooberry, SL; Sabat, M; Rieger, J; Brown, ML Structure-based discovery of a boronic acid bioisostere of combretastatin A-4. Chem Biol 12:1007-14 (2005) [PubMed] Article
More Info.:
Target
Name:
Tubulin polymerization-promoting protein
Synonyms:
TPPP | TPPP1 | TPPP_HUMAN | Tubulin | Tubulin polymerization-promoting protein
Type:
Protein
Mol. Mass.:
23706.03
Organism:
Homo sapiens (Human)
Description:
O94811
Residue:
219
Sequence:
MADKAKPAKAANRTPPKSPGDPSKDRAAKRLSLESEGAGEGAAASPELSALEEAFRRFAVHGDARATGREMHGKNWSKLCKDCQVIDGRNVTVTDVDIVFSKIKGKSCRTITFEQFQEALEELAKKRFKDKSSEEAVREVHRLIEGKAPIISGVTKAISSPTVSRLTDTTKFTGSHKERFDPSGKGKGKAGRVDLVDESGYVSGYKHAGTYDQKVQGGK