Reaction Details Report a problem with these data
Target
Neuropeptide Y receptor type 2
Ligand
BDBM29666
Substrate
n/a
Meas. Tech.
Fluorescence-based cell-based high-throughput dose response assay for agonists of NPY-Y2.
EC50
>35430±n/a nM
Citation
 PubChem, PC Fluorescence-based cell-based high-throughput dose response assay for agonists of NPY-Y2. PubChem Bioassay (2009)[AID] 
Target
Name:
Neuropeptide Y receptor type 2
Synonyms:
NPY-Y2 | NPY-Y2 receptor | NPY2-R | NPY2R | NPY2R_HUMAN | Neuropeptide Y receptor type 2 | Y2 receptor | neuropeptide Y receptor Y2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42734.65
Organism:
Homo sapiens (Human)
Description:
NPY-Y2 NPY2R HUMAN::P49146
Residue:
381
Sequence:
MGPIGAEADENQTVEEMKVEQYGPQTTPRGELVPDPEPELIDSTKLIEVQVVLILAYCSIILLGVIGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGPVLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKRISFLIIGLAWGISALLASPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSIYGTVYSLSSLLILYVLPLGIISFSYTRIWSKLKNHVSPGAANDHYHQRRQKTTKMLVCVVVVFAVSWLPLHAFQLAVDIDSQVLDLKEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSVTFKAKKNLEVRKNSGPNDSFTEATNV
  
Inhibitor
Name:
BDBM29666
Synonyms:
(9-Oxo-9H-acridin-10-yl)-acetic acid [1-(4-chloro-phenyl)-2,5-dimethyl-1H-pyrrol-3-ylmethylene]-hydrazide | MLS000566445 | N-[[1-(4-chlorophenyl)-2,5-dimethyl-3-pyrrolyl]methylideneamino]-2-(9-oxo-10-acridinyl)acetamide | N-[[1-(4-chlorophenyl)-2,5-dimethyl-pyrrol-3-yl]methyleneamino]-2-(9-ketoacridin-10-yl)acetamide | N-[[1-(4-chlorophenyl)-2,5-dimethyl-pyrrol-3-yl]methylideneamino]-2-(9-oxidanylideneacridin-10-yl)ethanamide | N-[[1-(4-chlorophenyl)-2,5-dimethylpyrrol-3-yl]methylideneamino]-2-(9-oxoacridin-10-yl)acetamide | SMR000175921 | cid_3116772
Type:
Small organic molecule
Emp. Form.:
C28H23ClN4O2
Mol. Mass.:
482.961
SMILES:
Cc1cc(C=NNC(=O)Cn2c3ccccc3c(=O)c3ccccc23)c(C)n1-c1ccc(Cl)cc1 |w:5.5|
Structure:
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