Reaction Details Report a problem with these data
Target
Protein Rev
Ligand
BDBM67439
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction
IC50
14833±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction PubChem Bioassay (2010)[AID] 
Target
Name:
Protein Rev
Synonyms:
Human immunodeficiency virus type 1 REV | REV_HV1H2 | rev
Type:
PROTEIN
Mol. Mass.:
13078.11
Organism:
Human immunodeficiency virus 1
Description:
ChEMBL_79479
Residue:
116
Sequence:
MAGRSGDSDEELIRTVRLIKLLYQSNPPPNPEGTRQARRNRRRRWRERQRQIHSISERILGTYLGRSAEPVPLQLPPLERLTLDCNEDCGTSGTQGVGSPQILVESPTVLESGTKE
  
Inhibitor
Name:
BDBM67439
Synonyms:
MLS001044354 | N-(2-phenazinyl)acetamide | N-Phenazin-2-yl-acetamide | N-phenazin-2-ylacetamide | N-phenazin-2-ylethanamide | SMR000424882 | cid_607082
Type:
Small organic molecule
Emp. Form.:
C14H11N3O
Mol. Mass.:
237.2566
SMILES:
CC(=O)Nc1ccc2nc3ccccc3nc2c1
Structure:
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