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Target
X-box-binding protein 1
Ligand
BDBM31063
Substrate
n/a
Meas. Tech.
XBP1 DR counterscreen for CHOP
IC50
10000±n/a nM
Citation
 PubChem, PC XBP1 DR counterscreen for CHOP PubChem Bioassay (2011)[AID] 
Target
Name:
X-box-binding protein 1
Synonyms:
TREB5 | XBP1 | XBP1_HUMAN | XBP2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
28704.14
Organism:
Homo sapiens (Human)
Description:
gi_47678753
Residue:
261
Sequence:
MVVVAAAPNPADGTPKVLLLSGQPASAAGAPAGQALPLMVPAQRGASPEAASGGLPQARKRQRLTHLSPEEKALRRKLKNRVAAQTARDRKKARMSELEQQVVDLEEENQKLLLENQLLREKTHGLVVENQELRQRLGMDALVAEEEAEAKGNEVRPVAGSAESAALRLRAPLQQVQAQLSPLQNISPWILAVLTLQIQSLISCWAFWTTWTQSCSSNALPQSLPAWRSSQRSTQKDPVPYQPPFLCQWGRHQPSWKPLMN
  
Inhibitor
Name:
BDBM31063
Synonyms:
2-(methylsulfonyl)-4-phenyl-6-(trifluoromethyl)pyrimidine | 2-mesyl-4-phenyl-6-(trifluoromethyl)pyrimidine | 2-methylsulfonyl-4-phenyl-6-(trifluoromethyl)pyrimidine | MLS000044644 | SMR000022588 | cid_3236803
Type:
Small organic molecule
Emp. Form.:
C12H9F3N2O2S
Mol. Mass.:
302.272
SMILES:
CS(=O)(=O)c1nc(cc(n1)C(F)(F)F)-c1ccccc1
Structure:
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