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Target
X-box-binding protein 1
Ligand
BDBM38993
Substrate
n/a
Meas. Tech.
XBP1 DR counterscreen for CHOP
IC50
2630±n/a nM
Citation
 PubChem, PC XBP1 DR counterscreen for CHOP PubChem Bioassay (2011)[AID] 
Target
Name:
X-box-binding protein 1
Synonyms:
TREB5 | XBP1 | XBP1_HUMAN | XBP2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
28704.14
Organism:
Homo sapiens (Human)
Description:
gi_47678753
Residue:
261
Sequence:
MVVVAAAPNPADGTPKVLLLSGQPASAAGAPAGQALPLMVPAQRGASPEAASGGLPQARKRQRLTHLSPEEKALRRKLKNRVAAQTARDRKKARMSELEQQVVDLEEENQKLLLENQLLREKTHGLVVENQELRQRLGMDALVAEEEAEAKGNEVRPVAGSAESAALRLRAPLQQVQAQLSPLQNISPWILAVLTLQIQSLISCWAFWTTWTQSCSSNALPQSLPAWRSSQRSTQKDPVPYQPPFLCQWGRHQPSWKPLMN
  
Inhibitor
Name:
BDBM38993
Synonyms:
(1Z,3Z)-1,4-bis(butylsulfonyl)buta-1,3-diene | MLS000085704 | SMR000020833 | cid_5286934
Type:
Small organic molecule
Emp. Form.:
C12H22O4S2
Mol. Mass.:
294.431
SMILES:
CCCCS(=O)(=O)\C=C/C=C\S(=O)(=O)CCCC
Structure:
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