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Target
X-box-binding protein 1
Ligand
BDBM67985
Substrate
n/a
Meas. Tech.
XBP1 DR counterscreen for CHOP
IC50
280±n/a nM
Citation
 PubChem, PC XBP1 DR counterscreen for CHOP PubChem Bioassay (2011)[AID] 
Target
Name:
X-box-binding protein 1
Synonyms:
TREB5 | XBP1 | XBP1_HUMAN | XBP2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
28704.14
Organism:
Homo sapiens (Human)
Description:
gi_47678753
Residue:
261
Sequence:
MVVVAAAPNPADGTPKVLLLSGQPASAAGAPAGQALPLMVPAQRGASPEAASGGLPQARKRQRLTHLSPEEKALRRKLKNRVAAQTARDRKKARMSELEQQVVDLEEENQKLLLENQLLREKTHGLVVENQELRQRLGMDALVAEEEAEAKGNEVRPVAGSAESAALRLRAPLQQVQAQLSPLQNISPWILAVLTLQIQSLISCWAFWTTWTQSCSSNALPQSLPAWRSSQRSTQKDPVPYQPPFLCQWGRHQPSWKPLMN
  
Inhibitor
Name:
BDBM67985
Synonyms:
5H-pyrimid[5,4-b]indol-4-yl-[(2,4,5-trimethoxybenzylidene)amino]amine | MLS000331873 | N-(5H-Pyrimido[5,4-b]indol-4-yl)-N'-[1-(2,4,5-trimethoxy-phenyl)-meth-(E)-ylidene]-hydrazine | N-[(2,4,5-trimethoxyphenyl)methylideneamino]-5H-pyrimido[5,4-b]indol-4-amine | SMR000221363 | cid_4887198
Type:
Small organic molecule
Emp. Form.:
C20H19N5O3
Mol. Mass.:
377.3966
SMILES:
COc1cc(OC)c(OC)cc1CN=Nc1ncnc2c3ccccc3[nH]c12 |w:14.15|
Structure:
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