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Target
X-box-binding protein 1
Ligand
BDBM68019
Substrate
n/a
Meas. Tech.
XBP1 DR counterscreen for CHOP
IC50
6310±n/a nM
Citation
 PubChem, PC XBP1 DR counterscreen for CHOP PubChem Bioassay (2011)[AID] 
Target
Name:
X-box-binding protein 1
Synonyms:
TREB5 | XBP1 | XBP1_HUMAN | XBP2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
28704.14
Organism:
Homo sapiens (Human)
Description:
gi_47678753
Residue:
261
Sequence:
MVVVAAAPNPADGTPKVLLLSGQPASAAGAPAGQALPLMVPAQRGASPEAASGGLPQARKRQRLTHLSPEEKALRRKLKNRVAAQTARDRKKARMSELEQQVVDLEEENQKLLLENQLLREKTHGLVVENQELRQRLGMDALVAEEEAEAKGNEVRPVAGSAESAALRLRAPLQQVQAQLSPLQNISPWILAVLTLQIQSLISCWAFWTTWTQSCSSNALPQSLPAWRSSQRSTQKDPVPYQPPFLCQWGRHQPSWKPLMN
  
Inhibitor
Name:
BDBM68019
Synonyms:
2-Chloro-3-phenylamino-[1,4]naphthoquinone | 2-anilino-3-chloro-1,4-naphthoquinone | 2-anilino-3-chloronaphthalene-1,4-dione | 2-chloranyl-3-phenylazanyl-naphthalene-1,4-dione | MLS000588884 | SMR000212533 | cid_14161
Type:
Small organic molecule
Emp. Form.:
C16H10ClNO2
Mol. Mass.:
283.709
SMILES:
ClC1=C(Nc2ccccc2)C(=O)c2ccccc2C1=O |c:1|
Structure:
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