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Target
Pituitary adenylate cyclase-activating polypeptide
Ligand
BDBM81760
Substrate
n/a
Ki
1000±n/a nM
Comments
PDSP_2373
Citation
 Robberecht, P; Gourlet, P; De Neef, P; Woussen-Colle, MC; Vandermeers-Piret, MC; Vandermeers, A; Christophe, J Receptor occupancy and adenylate cyclase activation in AR 4-2J rat pancreatic acinar cell membranes by analogs of pituitary adenylate cyclase-activating peptides amino-terminally shortened or modified at position 1, 2, 3, 20, or 21. Mol Pharmacol 42:347-55 (1992) [PubMed] 
Target
Name:
Pituitary adenylate cyclase-activating polypeptide
Synonyms:
Adcyap1 | PACAP | PACAP-27 | PACAP-38 | PACA_RAT | Pituitary adenylate cyclase-activating polypeptide
Type:
Enzyme Catalytic Domain
Mol. Mass.:
19565.66
Organism:
RAT
Description:
PACAP 0 RAT::P13589
Residue:
175
Sequence:
MTMCSGARLALLVYGIIMHNSVSCSPAAGLSFPGIRPEEEAYDQDGNPLQDFYDWDPPGAGSPASALRDAYALYYPADRRDVAHEILNEAYRKVLDQLSARKYLQSMVARGMGENLAAAAVDDRAPLTKRHSDGIFTDSYSRYRKQMAVKKYLAAVLGKRYKQRVKNKGRRIAYL
  
Inhibitor
Name:
BDBM81760
Synonyms:
[Des-His1,Glu3]PACAP-38
Type:
Small organic molecule
Emp. Form.:
C205H335N63O53S
Mol. Mass.:
4562.309
SMILES:
n/a
Structure:
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