Reaction Details Report a problem with these data
Target
P2Y purinoceptor 2
Ligand
BDBM81925
Substrate
n/a
Ki
4.3±n/a nM
Comments
PDSP_2952
Citation
Klotz, KN; Vogt, H; Tawfik-Schlieper, H Comparison of A1 adenosine receptors in brain from different species by radioligand binding and photoaffinity labelling. Naunyn Schmiedebergs Arch Pharmacol 343:196-201 (1991) [PubMed] Article
More Info.:
Target
Name:
P2Y purinoceptor 2
Synonyms:
ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | ADORA1 | P2RY2 | P2RY2_CRIGR | P2Y purinoceptor 2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
18813.49
Organism:
HAMSTER
Description:
ADENOSINE A1 ADORA1 HAMSTER::P58825
Residue:
166
Sequence:
VHRCLGVLRPLHSLRWGRARYARRVAAVVWVLVLACQAPVLYFVTTSVRGTRITCHDTSARELFSHFVAYSSVMLSLLFAVPFSVILVCYVLMARRLLKPAYGTTGGLPRAKRKSVRTIALVLAVFTLCFLPFHVTRTLYYSFRSLDLSCHTLNAINMAYKITRPL