Reaction Details Report a problem with these data
Target
kappa-type opioid receptor isoform 1
Ligand
BDBM81931
Substrate
n/a
Ki
0.1±n/a nM
Comments
PDSP_463
Citation
Benyhe, S; Varga, E; Hepp, J; Magyar, A; Borsodi, A; Wollemann, M Characterization of kappa 1 and kappa 2 opioid binding sites in frog (Rana esculenta) brain membrane preparation. Neurochem Res 15:899-904 (1990) [PubMed] Article
More Info.:
Target
Name:
kappa-type opioid receptor isoform 1
Synonyms:
OPIATE Kappa | OPRK1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42362.28
Organism:
Frog
Description:
F7A0F2
Residue:
375
Sequence:
MCFNLTMKKKKECCAPACPSSCFPNTSWLLGWDDHDNVSAYPDLPLNEGNHTSISPTISVIITAVYSMVFVVGLVGNALVMFVIIRYTKMKTATNIYIFNLALADALVTTTMPFQSTSFLMNSWPFGDVLCKIVVSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPLKAKCINICIWMLSSSVGISAIVLGGTKISDGSTECALQFPTHYWYWDTVMKMCVFIFAFIIPVFIITICYTLMILRLKSVRLLSGSREKDRNLRRITRLVLVVVAVFIVCWTPIHIFVLVEALVDVPQSIAVVSIYYFCIALGYTNSSLNPILYAFLDENFKRCFKDFCFPSKHRLDRQPNSRVGNTVQDPACNRHGSQKPV