Reaction Details Report a problem with these data
Target
Nicotinic acetylcholine receptor
Ligand
BDBM50060582
Substrate
n/a
Ki
3125±n/a nM
Comments
PDSP_632
Citation
 Lippiello, PM; Fernandes, KG The binding of L-[3H]nicotine to a single class of high affinity sites in rat brain membranes. Mol Pharmacol 29:448-54 (1986) [PubMed] 
Target
Name:
Nicotinic acetylcholine receptor
Synonyms:
Nicotinic acetylcholine receptor | n-AChR
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2478.99
Organism:
RAT
Description:
n-AChR 0 RAT::Q62594
Residue:
23
Sequence:
MTMALLGTLLLLALFGRSQGKNE
  
Inhibitor
Name:
BDBM50060582
Synonyms:
1,10-Bis(trimethyl ammonium)decane dibromide | 1,10-bis-(trimethyl ammonium) decane dibromide | CHEMBL1134 | DECAMETHONIUM | DECAMETHONIUM BROMIDE | Decamethonium Iodide | N,N,N'',N''-Tetramethyl-decane-1,10-diammonium; dibromide | N,N,N,N'',N'',N''-Hexamethyldecane-1,10-diammoniumdibromide | Syncurine | decane-1,10-bis(trimethylammonium bromide)
Type:
Small organic molecule
Emp. Form.:
C16H38N2
Mol. Mass.:
258.4852
SMILES:
C[N+](C)(C)CCCCCCCCCC[N+](C)(C)C
Structure:
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