Reaction Details Report a problem with these data
Target
Cholecystokinin
Ligand
BDBM82079
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_2674
Citation
 Van Dijk, A; Richards, JG; Trzeciak, A; Gillessen, D; Möhler, H Cholecystokinin receptors: biochemical demonstration and autoradiographical localization in rat brain and pancreas using [3H] cholecystokinin8 as radioligand. J Neurosci 4:1021-33 (1984) [PubMed] 
Target
Name:
Cholecystokinin
Synonyms:
CCKN_RAT | Cck
Type:
Enzyme Catalytic Domain
Mol. Mass.:
12844.29
Organism:
RAT
Description:
Cholecystokinin 0 RAT::P01355
Residue:
115
Sequence:
MKCGVCLCVVMAVLAAGALAQPVVPVEAVDPMEQRAEEAPRRQLRAVLRPDSEPRARLGALLARYIQQVRKAPSGRMSVLKNLQGLDPSHRISDRDYMGWMDFGRRSAEDYEYPS
  
Inhibitor
Name:
BDBM82079
Synonyms:
CAS_152221 | CCK4 | NSC_152221
Type:
Small organic molecule
Emp. Form.:
C35H46N6O8
Mol. Mass.:
678.7751
SMILES:
CCCCOC(=O)NC(=O)C(Cc1ccccc1)NC(=O)C(CC(O)=O)NC(=O)C(CC(C)C)NC(=O)C(N)Cc1c[nH]c2ccccc12
Structure:
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