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Target
Norepinephrine transporter
Ligand
BDBM82264
Substrate
n/a
Ki
432±n/a nM
Comments
PDSP_4115
Citation
 Codd, EE; Shank, RP; Schupsky, JJ; Raffa, RB Serotonin and norepinephrine uptake inhibiting activity of centrally acting analgesics: structural determinants and role in antinociception. J Pharmacol Exp Ther 274:1263-70 (1995) [PubMed] 
Target
Name:
Norepinephrine transporter
Synonyms:
n/a
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2082.45
Organism:
RAT
Description:
Norepinephrine transporter 0 RAT::Q9JIA2
Residue:
19
Sequence:
MLLARMKPQVQPELGGADQ
  
Inhibitor
Name:
BDBM82264
Synonyms:
CAS_19472 | CAS_27203-92-5 | NSC_19472 | Tramadol(+-) | Tramadol,(+) | Tramadol,(-)
Type:
Small organic molecule
Emp. Form.:
C13H18N3
Mol. Mass.:
216.3016
SMILES:
C1CN=C(N1)[NH2+]c1cccc2CCCCc12 |c:2|
Structure:
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