Reaction Details
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Report a problem with these dataTarget
Somatostatin receptor type 4
Ligand
BDBM82463
Substrate
n/a
Ki
63.09±n/a nM
Comments
PDSP_1033
Citation
Hoyer, D; Lübbert, H; Bruns, C Molecular pharmacology of somatostatin receptors. Naunyn Schmiedebergs Arch Pharmacol 350:441-53 (1994) [PubMed] Article More Info.:
Target
Name:
Somatostatin receptor type 4
Synonyms:
SS-4-R | SS4-R | SS4R | SSR4_MOUSE | Smstr4 | Sstr4
Type:
PROTEIN
Mol. Mass.:
41937.48
Organism:
Mus musculus
Description:
ChEMBL_833920
Residue:
385
Sequence:
MNAPATLPPGVEDTTWTPGINASWAPDEEEEDAMGSDGTGTAGMVTIQCIYALVCLVGLVGNALVIFVILRYAKMKTATNIYLLNLAVADELFMLSVPFARSAAALRHWPFGAVLCRAVLSVDGLNMFTSVFCLTVLSVDRYVAVVHPLATATYRRPSVAKLINLGVWLASLLVTLPIAVFADTRPARGGEAVACNLHWPHPAWSAVFVIYTFLLGFLPPVLAIGLCYLLIVGKMRAVALAGGWQQRRRSEKKITRLVLMVVTVFVLCWMPFYVVQLLNLFVTSLDATVNHVSLILSYANSCANPILYGFLSDNFRRSFQRVLCLRCCLLETTGGAEEEPLDYYATALKSRGGAGCICPPLPCQQEPVQAEPGCKQVPFTKTTTF
Inhibitor
Name:
BDBM82463
Synonyms:
Cyclo[L-Trp-D-Trp-L-Lys-L-Thr-L-Phe-(7-amino*heptanoyl-L-Phe-)] | L-362,855 | L-362855
Type:
Small organic molecule
Emp. Form.:
C57H70N10O8
Mol. Mass.:
1023.2279
SMILES:
C[C@@H](O)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)CCCCCCNC(=O)[C@H](Cc2ccccc2)NC1=O
Structure:
