Reaction Details
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5-hydroxytryptamine receptor 1B
Ligand
BDBM81498
Substrate
n/a
Ki
10±n/a nM
Comments
PDSP_1643
Citation
Boess, FG; Martin, IL Molecular biology of 5-HT receptors. Neuropharmacology 33:275-317 (1994) [PubMed] Article More Info.:
Target
Name:
5-hydroxytryptamine receptor 1B
Synonyms:
5-HT1B | 5-hydroxytryptamine receptor 1B (5HT1B) | 5HT1B_MOUSE | 5ht1b | Htr1b
Type:
Enzyme
Mol. Mass.:
43090.29
Organism:
Mus musculus (Mouse)
Description:
P28334
Residue:
386
Sequence:
MEEQGIQCAPPPPAASQTGVPLTNLSHNCSADGYIYQDSIALPWKVLLVALLALITLATTLSNAFVIATVYRTRKLHTPANYLIASLAVTDLLVSILVMPISTMYTVTGRWTLGQVVCDFWLSSDITCCTASIMHLCVIALDRYWAITDAVEYSAKRTPKRAAIMIVLVWVFSISISLPPFFWRQAKAEEEMLDCFVNTDHVLYTVYSTVGAFYLPTLLLIALYGRIYVEARSRILKQTPNKTGKRLTRAQLITDSPGSTSSVTSINSRAPDVPSESGSPVYVNQVKVRVSDALLEKKKLMAARERKATKTLGIILGAFIVCWLPFFIISLVMPICKDACWFHMAIFDFFNWLGYLNSLINPIIYTMSNEDFKQAFHKLIRFKCAG
Inhibitor
Name:
BDBM81498
Synonyms:
5-Methoxy-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole(RU-24969) | CAS_108028 | CHEMBL18785 | NSC_108028 | RU 24969
Type:
Small organic molecule
Emp. Form.:
C14H16N2O
Mol. Mass.:
228.2896
SMILES:
COc1ccc2[nH]cc(C3=CCNCC3)c2c1 |t:9|
Structure:
