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Target
G-protein coupled receptor 52
Ligand
BDBM50252099
Substrate
n/a
Meas. Tech.
ChEBML_1684383
EC50
23±n/a nM
Citation
 Tokumaru, K; Ito, Y; Nomura, I; Nakahata, T; Shimizu, Y; Kurimoto, E; Aoyama, K; Aso, K Design, synthesis, and pharmacological evaluation of 4-azolyl-benzamide derivatives as novel GPR52 agonists. Bioorg Med Chem 25:3098-3115 (2017) [PubMed]  Article 
Target
Name:
G-protein coupled receptor 52
Synonyms:
GPR52 | GPR52_HUMAN | Probable G-protein coupled receptor 52
Type:
PROTEIN
Mol. Mass.:
41366.15
Organism:
Homo sapiens (Human)
Description:
ChEMBL_108391
Residue:
361
Sequence:
MNESRWTEWRILNMSSGIVNVSERHSCPLGFGHYSVVDVCIFETVVIVLLTFLIIAGNLTVIFVFHCAPLLHHYTTSYFIQTMAYADLFVGVSCLVPTLSLLHYSTGVHESLTCQVFGYIISVLKSVSMACLACISVDRYLAITKPLSYNQLVTPCRLRICIILIWIYSCLIFLPSFFGWGKPGYHGDIFEWCATSWLTSAYFTGFIVCLLYAPAAFVVCFTYFHIFKICRQHTKEINDRRARFPSHEVDSSRETGHSPDRRYAMVLFRITSVFYMLWLPYIIYFLLESSRVLDNPTLSFLTTWLAISNSFCNCVIYSLSNSVFRLGLRRLSETMCTSCMCVKDQEAQEPKPRKRANSCSI
  
Inhibitor
Name:
BDBM50252099
Synonyms:
CHEMBL4087237
Type:
Small organic molecule
Emp. Form.:
C20H17F4N3O
Mol. Mass.:
391.3621
SMILES:
Cc1cc(ccc1C(N)=O)-c1cc(Cc2cc(F)cc(c2)C(F)(F)F)nn1C
Structure:
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