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Target
G-protein coupled receptor 52
Ligand
BDBM50252092
Substrate
n/a
Meas. Tech.
ChEBML_1684415
EC50
71±n/a nM
Citation
 Tokumaru, K; Ito, Y; Nomura, I; Nakahata, T; Shimizu, Y; Kurimoto, E; Aoyama, K; Aso, K Design, synthesis, and pharmacological evaluation of 4-azolyl-benzamide derivatives as novel GPR52 agonists. Bioorg Med Chem 25:3098-3115 (2017) [PubMed]  Article 
Target
Name:
G-protein coupled receptor 52
Synonyms:
G-protein coupled receptor 52 | GPR52_MOUSE | Gpr52
Type:
PROTEIN
Mol. Mass.:
41353.59
Organism:
Mus musculus
Description:
ChEMBL_117396
Residue:
361
Sequence:
MNESRWTEWRILNMSSSIVNVSEHHSCPLGFGHYSVEDVCIFETVVIVLLTFLIISGNLTVIFVFHCAPLLHHYTTSYFIQTMAYADLLVGVTCLVPTLSLLHYSTGVHESLTCQVFGYIISVLKSVSMACLACISVDRYLAITKPLSYNQLVTPCRLRICIIMIWIYSCLIFLPSFFGWGKPGYHGDIFEWCATSWLTSAYFTCFIVCLLYAPAALVVCFTYFHIFKICRQHTKEINDRRARFPSHEVEASREAGHSPDRRYAMVLFRITSVFYMLWLPYIIYFLLESSRVLDNPTLSFLTTWLAISNSFCNCVIYSLSNSVFRLGLRRLSETMCTSCVCAKDQEAQDPKPRRRANSCSI
  
Inhibitor
Name:
BDBM50252092
Synonyms:
CHEMBL4082756
Type:
Small organic molecule
Emp. Form.:
C19H16F4N4O
Mol. Mass.:
392.3502
SMILES:
Cc1nc(Cc2cc(F)cc(c2)C(F)(F)F)nn1-c1ccc(C(N)=O)c(C)c1
Structure:
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