Reaction Details Report a problem with these data
Target
Adenosine receptor A3
Ligand
BDBM50266662
Substrate
n/a
Meas. Tech.
ChEMBL_1701162 (CHEMBL4052144)
Ki
65±n/a nM
Citation
 Petrelli, R; Scortichini, M; Kachler, S; Boccella, S; Cerchia, C; Torquati, I; Del Bello, F; Salvemini, D; Novellino, E; Luongo, L; Maione, S; Jacobson, KA; Lavecchia, A; Klotz, KN; Cappellacci, L Exploring the Role of N J Med Chem 60:4327-4341 (2017) [PubMed]  Article 
Target
Name:
Adenosine receptor A3
Synonyms:
Adenosine A3 receptor | AA3R_RAT | Adora3 | Adenosine receptor A2a and A3
Type:
PROTEIN
Mol. Mass.:
36643.73
Organism:
Rat
Description:
ChEMBL_479910
Residue:
320
Sequence:
MKANNTTTSALWLQITYITMEAAIGLCAVVGNMLVIWVVKLNRTLRTTTFYFIVSLALADIAVGVLVIPLAIAVSLEVQMHFYACLFMSCVLLVFTHASIMSLLAIAVDRYLRVKLTVRYRTVTTQRRIWLFLGLCWLVSFLVGLTPMFGWNRKVTLELSQNSSTLSCHFRSVVGLDYMVFFSFITWILIPLVVMCIIYLDIFYIIRNKLSQNLTGFRETRAFYGREFKTAKSLFLVLFLFALCWLPLSIINFVSYFNVKIPEIAMCLGILLSHANSMMNPIVYACKIKKFKETYFVILRACRLCQTSDSLDSNLEQTTE
  
Inhibitor
Name:
BDBM50266662
Synonyms:
CHEMBL4087306
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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