Reaction Details Report a problem with these data
Target
P2Y purinoceptor 2
Ligand
BDBM50271600
Substrate
n/a
Meas. Tech.
ChEMBL_1711179 (CHEMBL4121228)
Ki
83±n/a nM
Citation
 Conroy, S; Kindon, ND; Glenn, J; Stoddart, LA; Lewis, RJ; Hill, SJ; Kellam, B; Stocks, MJ Synthesis and Evaluation of the First Fluorescent Antagonists of the Human P2Y J Med Chem 61:3089-3113 (2018) [PubMed]  Article 
Target
Name:
P2Y purinoceptor 2
Synonyms:
ATP receptor | P2RU1 | P2RY2 | P2RY2_HUMAN | P2U purinoceptor 1 | P2U1 | P2Y purinoceptor 2 | P2Y2 | Purinergic receptor | Purinergic receptor P2Y2
Type:
PROTEIN
Mol. Mass.:
42299.21
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1455361
Residue:
377
Sequence:
MAADLGPWNDTINGTWDGDELGYRCRFNEDFKYVLLPVSYGVVCVPGLCLNAVALYIFLCRLKTWNASTTYMFHLAVSDALYAASLPLLVYYYARGDHWPFSTVLCKLVRFLFYTNLYCSILFLTCISVHRCLGVLRPLRSLRWGRARYARRVAGAVWVLVLACQAPVLYFVTTSARGGRVTCHDTSAPELFSRFVAYSSVMLGLLFAVPFAVILVCYVLMARRLLKPAYGTSGGLPRAKRKSVRTIAVVLAVFALCFLPFHVTRTLYYSFRSLDLSCHTLNAINMAYKVTRPLASANSCLDPVLYFLAGQRLVRFARDAKPPTGPSPATPARRRLGLRRSDRTDMQRIEDVLGSSEDSRRTESTPAGSENTKDIRL
  
Inhibitor
Name:
BDBM50271600
Synonyms:
CHEMBL4086462
Type:
Small organic molecule
Emp. Form.:
C25H23Cl2N2Na4O13P3S
Mol. Mass.:
847.307
SMILES:
n/a
Structure:
Search PDB for entries with ligand similarity: