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Target
Prostaglandin E2 receptor EP2 subtype
Ligand
BDBM50454063
Substrate
n/a
Meas. Tech.
ChEMBL_1751764 (CHEMBL4186524)
EC50
0.110000±n/a nM
Citation
 Kinoshita, A; Higashino, M; Yoshida, K; Aratani, Y; Kakuuchi, A; Hanada, K; Takeda, H; Naganawa, A; Matsuya, H; Ohmoto, K Synthesis and evaluation of a potent, well-balanced EP Bioorg Med Chem 26:200-214 (2018) [PubMed]  Article 
Target
Name:
Prostaglandin E2 receptor EP2 subtype
Synonyms:
PGE receptor EP2 subtype | Prostaglandin E2 | Prostanoid EP2 Receptor | PE2R2_HUMAN | PTGER2 | Prostaglandin E2 receptor | Prostaglandin E2 receptor EP4 subtype
Type:
Enzyme
Mol. Mass.:
39775.71
Organism:
Human
Description:
P43116
Residue:
358
Sequence:
MGNASNDSQSEDCETRQWLPPGESPAISSVMFSAGVLGNLIALALLARRWRGDVGCSAGRRSSLSLFHVLVTELVFTDLLGTCLISPVVLASYARNQTLVALAPESRACTYFAFAMTFFSLATMLMLFAMALERYLSIGHPYFYQRRVSRSGGLAVLPVIYAVSLLFCSLPLLDYGQYVQYCPGTWCFIRHGRTAYLQLYATLLLLLIVSVLACNFSVILNLIRMHRRSRRSRCGPSLGSGRGGPGARRRGERVSMAEETDHLILLAIMTITFAVCSLPFTIFAYMNETSSRKEKWDLQALRFLSINSIIDPWVFAILRPPVLRLMRSVLCCRISLRTQDATQTSCSTQSDASKQADL
  
Inhibitor
Name:
BDBM50454063
Synonyms:
CHEMBL4205480
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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