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Target
5-hydroxytryptamine receptor 5A
Ligand
BDBM50456729
Substrate
n/a
Meas. Tech.
ChEMBL_1757988 (CHEMBL4192996)
Ki
>10000±n/a nM
Citation
 Lin, Z; Smith, MD; Concepcion, GP; Haygood, MG; Olivera, BM; Light, A; Schmidt, EW Modulating the Serotonin Receptor Spectrum of Pulicatin Natural Products. J Nat Prod 80:2360-2370 (2017) [PubMed]  Article 
Target
Name:
5-hydroxytryptamine receptor 5A
Synonyms:
5-HT-5 | 5-HT-5A | 5-hydroxytryptamine receptor 5 (5-HT5) | 5-hydroxytryptamine receptor 5A (5-HT5A) | 5HT5A_HUMAN | HTR5A | Serotonin (5-HT) receptor | Serotonin receptor 5A
Type:
Enzyme
Mol. Mass.:
40266.25
Organism:
Homo sapiens (Human)
Description:
P47898
Residue:
357
Sequence:
MDLPVNLTSFSLSTPSPLETNHSLGKDDLRPSSPLLSVFGVLILTLLGFLVAATFAWNLLVLATILRVRTFHRVPHNLVASMAVSDVLVAALVMPLSLVHELSGRRWQLGRRLCQLWIACDVLCCTASIWNVTAIALDRYWSITRHMEYTLRTRKCVSNVMIALTWALSAVISLAPLLFGWGETYSEGSEECQVSREPSYAVFSTVGAFYLPLCVVLFVYWKIYKAAKFRVGSRKTNSVSPISEAVEVKDSAKQPQMVFTVRHATVTFQPEGDTWREQKEQRAALMVGILIGVFVLCWIPFFLTELISPLCSCDIPAIWKSIFLWLGYSNSFFNPLIYTAFNKNYNSAFKNFFSRQH
  
Inhibitor
Name:
BDBM50456729
Synonyms:
CHEMBL4202582
Type:
Small organic molecule
Emp. Form.:
C13H14N2OS
Mol. Mass.:
246.328
SMILES:
C[C@@H]1SC(=N[C@H]1CO)c1c[nH]c2ccccc12 |r,c:3|
Structure:
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