Reaction Details Report a problem with these data
Target
Cytosol aminopeptidase [435-519]
Ligand
BDBM50022748
Substrate
n/a
Meas. Tech.
ChEMBL_1759797 (CHEMBL4194805)
Ki
22±n/a nM
Citation
 Amin, SA; Adhikari, N; Jha, T Design of Aminopeptidase N Inhibitors as Anti-cancer Agents. J Med Chem 61:6468-6490 (2018) [PubMed]  Article 
Target
Name:
Cytosol aminopeptidase [435-519]
Synonyms:
3.4.11.1 | AMPL_PIG | LAP3 | Leucine aminopeptidase
Type:
PROTEIN
Mol. Mass.:
9577.41
Organism:
Sus scrofa
Description:
ChEMBL_116728
Residue:
85
Sequence:
FEHYTKQIVDCQLADVNNIGKYRSAGACTAAAFLKEFVTHPKWAHLDIAGVMTNKDEVPYLRKGMAGRPTRTLIEFLLRFSQDSA
  
Inhibitor
Name:
BDBM50022748
Synonyms:
2-Amino-4-methyl-pentane-1-thiol | CHEMBL69349
Type:
Small organic molecule
Emp. Form.:
C6H15NS
Mol. Mass.:
133.255
SMILES:
CC(C)C[C@@H](N)CS
Structure:
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