Reaction Details Report a problem with these data
Target
ADP-ribose glycohydrolase MACROD2
Ligand
BDBM50460478
Substrate
n/a
Meas. Tech.
ChEBML_1769550
Kd
150±n/a nM
Citation
Zhang, Y; Jumppanen, M; Maksimainen, MM; Auno, S; Awol, Z; Ghemtio, L; Venkannagari, H; Lehtiö, L; Yli-Kauhaluoma, J; Xhaard, H; Boije Af Gennäs, G Adenosine analogs bearing phosphate isosteres as human MDO1 ligands. Bioorg Med Chem 26:1588-1597 (2018) [PubMed] Article
More Info.:
Target
Name:
ADP-ribose glycohydrolase MACROD2
Synonyms:
3.2.2.- | 3.5.1.- | ADP-ribose glycohydrolase MACROD2 | C20orf133 | MACD2_HUMAN | MACRO domain-containing protein 2 | MACROD2 | O-acetyl-ADP-ribose deacetylase MACROD2 | [Protein ADP-ribosylaspartate] hydrolase MACROD2 | [Protein ADP-ribosylglutamate] hydrolase MACROD2
Type:
PROTEIN
Mol. Mass.:
47383.93
Organism:
Homo sapiens
Description:
ChEMBL_117875
Residue:
425
Sequence:
MYPSNKKKKVWREEKERLLKMTLEERRKEYLRDYIPLNSILSWKEEMKGKGQNDEENTQETSQVKKSLTEKVSLYRGDITLLEVDAIVNAANASLLGGGGVDGCIHRAAGPCLLAECRNLNGCDTGHAKITCGYDLPAKYVIHTVGPIARGHINGSHKEDLANCYKSSLKLVKENNIRSVAFPCISTGIYGFPNEPAAVIALNTIKEWLAKNHHEVDRIIFCVFLEVDFKIYKKKMNEFFSVDDNNEEEEDVEMKEDSDENGPEEKQSVEEMEEQSQDADGVNTVTVPGPASEEAVEDCKDEDFAKDENITKGGEVTDHSVRDQDHPDGQENDSTKNEIKIETESQSSYMETEELSSNQEDAVIVEQPEVIPLTEDQEEKEGEKAPGEDTPRMPGKSEGSSDLENTPGPDAGAQDEAKEQRNGTK