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Target
D(1A) dopamine receptor
Ligand
BDBM50461411
Substrate
n/a
Meas. Tech.
ChEMBL_1771299 (CHEMBL4223411)
Ki
128±n/a nM
Citation
 Omran, A; Eslamimehr, S; Crider, AM; Neumann, WL Synthesis of 3-(3-hydroxyphenyl)pyrrolidine dopamine D Bioorg Med Chem Lett 28:1897-1902 (2018) [PubMed]  Article 
Target
Name:
D(1A) dopamine receptor
Synonyms:
DA D1 receptor | DOPAMINE D1 | DRD1 | DRD1_HUMAN | Dopamine D1 receptor | Dopamine D1 receptor (D1R) | Dopamine D1A
Type:
Enzyme
Mol. Mass.:
49303.43
Organism:
Homo sapiens (Human)
Description:
P21728
Residue:
446
Sequence:
MRTLNTSAMDGTGLVVERDFSVRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTNFFVISLAVSDLLVAVLVMPWKAVAEIAGFWPFGSFCNIWVAFDIMCSTASILNLCVISVDRYWAISSPFRYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPTSPSDGNATSLAETIDNCDSSLSRTYAISSSVISFYIPVAIMIVTYTRIYRIAQKQIRRIAALERAAVHAKNCQTTTGNGKPVECSQPESSFKMSFKRETKVLKTLSVIMGVFVCCWLPFFILNCILPFCGSGETQPFCIDSNTFDVFVWFGWANSSLNPIIYAFNADFRKAFSTLLGCYRLCPATNNAIETVSINNNGAAMFSSHHEPRGSISKECNLVYLIPHAVGSSEDLKKEEAAGIARPLEKLSPALSVILDYDTDVSLEKIQPITQNGQHPT
  
Inhibitor
Name:
BDBM50461411
Synonyms:
CHEMBL4229178
Type:
Small organic molecule
Emp. Form.:
C20H33NO
Mol. Mass.:
303.4821
SMILES:
CCCCCCCCCCN1CCC(C1)c1cccc(O)c1
Structure:
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