Reaction Details Report a problem with these data
Target
14-3-3 protein gamma
Ligand
BDBM50102295
Substrate
n/a
Meas. Tech.
ChEMBL_1772679 (CHEMBL4229671)
IC50
16400±n/a nM
Citation
Stevers, LM; Sijbesma, E; Botta, M; MacKintosh, C; Obsil, T; Landrieu, I; Cau, Y; Wilson, AJ; Karawajczyk, A; Eickhoff, J; Davis, J; Hann, M; O'Mahony, G; Doveston, RG; Brunsveld, L; Ottmann, C Modulators of 14-3-3 Protein-Protein Interactions. J Med Chem 61:3755-3778 (2018) [PubMed] Article
More Info.:
Target
Name:
14-3-3 protein gamma
Synonyms:
1433G_HUMAN | YWHAG | tyrosine 3-monooxygenase/tryptophan 5-monooxygenase activation protein, gamma polypeptide
Type:
Enzyme Catalytic Domain
Mol. Mass.:
28289.17
Organism:
Homo sapiens (Human)
Description:
gi_21464101
Residue:
247
Sequence:
MVDREQLVQKARLAEQAERYDDMAAAMKNVTELNEPLSNEERNLLSVAYKNVVGARRSSWRVISSIEQKTSADGNEKKIEMVRAYREKIEKELEAVCQDVLSLLDNYLIKNCSETQYESKVFYLKMKGDYYRYLAEVATGEKRATVVESSEKAYSEAHEISKEHMQPTHPIRLGLALNYSVFYYEIQNAPEQACHLAKTAFDDAIAELDTLNEDSYKDSTLIMQLLRDNLTLWTSDQQDDDGGEGNN