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Target
Protein kinase domain-containing protein
Ligand
BDBM50265025
Substrate
n/a
Meas. Tech.
ChEMBL_900187 (CHEMBL3047469)
IC50
440±n/a nM
Citation
  TBA Med Chem Res 21:681-693 (2012)    Article 
Target
Name:
Protein kinase domain-containing protein
Synonyms:
Putative uncharacterized protein pk7
Type:
PROTEIN
Mol. Mass.:
37967.83
Organism:
Plasmodium falciparum
Description:
ChEMBL_496798
Residue:
320
Sequence:
MKDILSNYSNLIYLNKYVKEKDKYINDYRIIRTLNQGKFNKIILCEKDNKFYALKKYEKSLLEKKRDFTKSNNDKISIKSKYDDFKNELQIITDIKNEYCLTCEGIITNYDEVYIIYEYMENDSILKFDEYFFVLDKNYTCFIPIQVIKCIIKSVLNSFSYIHNEKNICHRDVKPSNILMDKNGRVKLSDFGESEYMVDKKIKGSRGTYEFMPPEFFSNESSYNGAKVDIWSLGICLYVMFYNVVPFSLKISLVELFNNIRTKNIEYPLDRNHFLYPLTNKKSTCSNNFLSNEDIDFLKLFLRKNPAERITSEDALVTAK
  
Inhibitor
Name:
BDBM50265025
Synonyms:
(S)-4-(6-(1-hydroxypropan-2-ylamino)imidazo[1,2-b]pyridazin-3-yl)benzonitrile | CHEMBL496538
Type:
Small organic molecule
Emp. Form.:
C16H15N5O
Mol. Mass.:
293.3232
SMILES:
C[C@@H](CO)Nc1ccc2ncc(-c3ccc(cc3)C#N)n2n1 |r|
Structure:
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