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Target
cAMP-specific 3',5'-cyclic phosphodiesterase 4A
Ligand
BDBM15296
Substrate
n/a
Meas. Tech.
ChEMBL_909208 (CHEMBL3054104)
Ki
4670±n/a nM
Citation
  TBA Med Chem Res 17:587-603 (2008)    Article 
Target
Name:
cAMP-specific 3',5'-cyclic phosphodiesterase 4A
Synonyms:
3.1.4.53 | PDE4A | PDE4A_CAVPO
Type:
PROTEIN
Mol. Mass.:
13503.64
Organism:
Cavia porcellus
Description:
ChEMBL_106603
Residue:
117
Sequence:
PWLVGWWDQFKRMLNRELTHLSEMSRSGNQVSEYISTTFLDKQNEVEIPSPTMKDREPQEAPRQRPCQQLPPPVPHLQPMSQITGVKRLSHNSGLNNASIPRFGVKTDQEELLAQEL
  
Inhibitor
Name:
BDBM15296
Synonyms:
6-methyl-2-oxo-5-(pyridin-4-yl)-1,2-dihydropyridine-3-carbonitrile | 6-methyl-2-oxo-5-pyridin-4-yl-1H-pyridine-3-carbonitrile | CHEMBL189 | Milrinone | Primacor | US9242982, Milrinone | US9249139, Milrinone
Type:
Small organic molecule
Emp. Form.:
C12H9N3O
Mol. Mass.:
211.2194
SMILES:
Cc1[nH]c(=O)c(cc1-c1ccncc1)C#N
Structure:
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