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Target
Protein ultraspiracle
Ligand
BDBM50128305
Substrate
n/a
Meas. Tech.
ChEMBL_925682 (CHEMBL3069808)
EC50
16596±n/a nM
Citation
 Soin, T; Swevers, L; Kotzia, G; Iatrou, K; Janssen, CR; Rougé, P; Harada, T; Nakagawa, Y; Smagghe, G Comparison of the activity of non-steroidal ecdysone agonists between dipteran and lepidopteran insects, using cell-based EcR reporter assays. Pest Manag Sci 66:1215-29 (2010) [PubMed]  Article 
Target
Name:
Protein ultraspiracle
Synonyms:
Cf1 | Chorion factor 1 | NR2B4 | Nuclear receptor subfamily 2 group B member 4 | USP_DROME | XR2C | usp
Type:
PROTEIN
Mol. Mass.:
55254.53
Organism:
Drosophila melanogaster
Description:
ChEMBL_106725
Residue:
508
Sequence:
MDNCDQDASFRLSHIKEEVKPDISQLNDSNNSSFSPKAESPVPFMQAMSMVHVLPGSNSASSNNNSAGDAQMAQAPNSAGGSAAAAVQQQYPPNHPLSGSKHLCSICGDRASGKHYGVYSCEGCKGFFKRTVRKDLTYACRENRNCIIDKRQRNRCQYCRYQKCLTCGMKREAVQEERQRGARNAAGRLSASGGGSSGPGSVGGSSSQGGGGGGGVSGGMGSGNGSDDFMTNSVSRDFSIERIIEAEQRAETQCGDRALTFLRVGPYSTVQPDYKGAVSALCQVVNKQLFQMVEYARMMPHFAQVPLDDQVILLKAAWIELLIANVAWCSIVSLDDGGAGGGGGGLGHDGSFERRSPGLQPQQLFLNQSFSYHRNSAIKAGVSAIFDRILSELSVKMKRLNLDRRELSCLKAIILYNPDIRGIKSRAEIEMCREKVYACLDEHCRLEHPGDDGRFAQLLLRLPALRSISLKCQDHLFLFRITSDRPLEELFLEQLEAPPPPGLAMKLE
  
Inhibitor
Name:
BDBM50128305
Synonyms:
3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenzoyl)-2-(1,1-dimethylethyl)hydrazide | CHEMBL55772 | N'-(tert-butyl)-N'-(3,5-dimethylbenzoyl)-3-methoxy-2-methylbenzohydrazide | N'-tert-butyl-N'-(3,5-dimethylbenzoyl)-3-methoxy-2-methylbenzohydrazide | N-tert-butyl-N'-(3-methoxy-o-toluoyl)-3,5-xylohydrazide | methoxyfenozide
Type:
Small organic molecule
Emp. Form.:
C22H28N2O3
Mol. Mass.:
368.4693
SMILES:
COc1cccc(C(=O)NN(C(=O)c2cc(C)cc(C)c2)C(C)(C)C)c1C
Structure:
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