Reaction Details Report a problem with these data
Target
Ecdysone receptor/Protein ultraspiracle homolog
Ligand
BDBM50178988
Substrate
n/a
Meas. Tech.
ChEMBL_927367 (CHEMBL3072567)
Ki
0.501187±n/a nM
Citation
Tohidi-Esfahani, D; Lawrence, MC; Graham, LD; Hannan, GN; Simpson, AM; Hill, RJ Isoforms of the heteropteran Nezara viridula ecdysone receptor: protein characterisation, RH5992 insecticide binding and homology modelling. Pest Manag Sci 67:1457-67 (2011) [PubMed] Article
More Info.:
Target
Name:
Ecdysone receptor/Protein ultraspiracle homolog
Synonyms:
Ecdysone receptor
Type:
n/a
Mol. Mass.:
n/a
Description:
ASSAY_ID of ChEMBL is 927367
Components:
This complex has 2 components.
Component 1
Name:
Ecdysone receptor
Synonyms:
n/a
Type:
PROTEIN
Mol. Mass.:
57629.46
Organism:
Choristoneura fumiferana
Description:
ChEMBL_65458
Residue:
513
Sequence:
MDLKHEVAYRGVLPGQVKAEPGVHNGQVNGHVRDWMAGGAGANSPSPGAVAQPQPNNGYSSPLSSGSYGPYSPNGKIGREELSPASSINGCSTDGEARRQKKGPAPRQQEELCLVCGDRASGYHYNALTCEGCKGFFRRSVTKNAVYICKFGHACEMDMYMRRKCQECRLKKCLAVGMRPECVVPETQCAMKRKEKKAQKEKDKLPVSTTTVDDHMPPIMQCEPPPPEAARIHEVVPRFLSDKLLETNRQKNIPQLTANQQFLIARLIWYQDGYEQPSDEDLKRITQTWQQADDENEESDTPFRQITEMTILTVQLIVEFAKGLPGFAKISQPDQITLLKACSSEVMMLRVARRYDAASDSVLFANNQAYTRDNYRKAGMAYVIEDLLHFCRCMYSMALDNIHYALLTAVVIFSDRPGLEQPQLVEEIQRYYLNTLRIYILNQLSGSARSSVIYGKILSILSELRTLGMQNSNMCISLKLKNRKLPPFLEEIWDVADMSHTQPPPILESPTNL
Component 2
Name:
Protein ultraspiracle homolog
Synonyms:
NR2B4 | Nuclear receptor subfamily 2 group B member 4 | Protein ultraspiracle homolog | USP | USP_CHOFU
Type:
PROTEIN
Mol. Mass.:
53145.42
Organism:
Choristoneura fumiferana
Description:
ChEMBL_106724
Residue:
472
Sequence:
MSSVAKKDKPTMSVTALINWARPAPPGPPQPQSASPAPAAMLQQLPTQSMQSLNHIPTVDCSLDMQWLNLEPGFMSPMSPPEMKPDTAMLDGLRDDATSPPNFKNYPPNHPLSGSKHLCSICGDRASGKHYGVYSCEGCKGFFKRTVRKDLSYACREERNCIIDKRQRNRCQYCRYQKCLACGMKREAVQEERQRNARGAEDAHPSSSVQVSDELSIERLTEMESLVADPSEEFQFLRVGPDSNVPPRYRAPVSSLCQIGNKQIAALVVWARDIPHFGQLELDDQVVLIKASWNELLLFAIAWRSMEYLEDERENGDGTRSTTQPQLMCLMPGMTLHRNSAQQAGVGAIFDRVLSELSLKMRTLRMDQAEYVALKAIVLLNPDVKGLKNRQEVDVLREKMFSCLDDYCRRSRSNEEGRFASLLLRLPALRSISLKSFEHLYFFHLVAEGSISGYIREALRNHAPPIDVNAMM